X-ray Structures of Succinimidyl Halobenzoates


X-ray Structures of Succinimidyl Halobenzoates

Mamat, C.; Weiss, D.-H.; Köckerling, M.

The crystal and molecular structures of five succinimidyl halobenzoates are reported. Corresponding derivatives with the respective halo-radionuclide (18F, 76Br, 123I/124I/125I/131I) were prepared and used for the radiolabeling of biologically active (macro-)molecules (peptides, proteins, antibodies) under mild labeling conditions. All compounds crystalized from petroleum ether/ethyl acetate mixtures.

Keywords: building block; radiolabeling; [18F]SFB; SIB; SBrB

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Publ.-Id: 25104