Design and synthesis of affine and selective histone deacetylase 1/2 inhibitors for imaging with PET

Publication

• O. Clauß, L. Schäker-Hübner, B. Wenzel, M. Toussaint, W. Deuther-Conrad, D. Gündel, R. Teodoro, S. Dukic-Stefanovic, F.-A. Ludwig, K. Kopka, P. Brust, F. K. Hansen, M. Scheunemann; Development and biological evaluation of the first highly potent and specific benzamide-based radiotracer [¹⁸F]BA3 for imaging histone deacetylases 1 and 2 in brain; Pharmaceuticals (2022). doi.org/10.3390/ph15030324