Publications of Institute of Radiopharmaceutical Cancer Research
409 Publications2019
Current management of pheochromocytoma/paraganglioma: A guide for the practicing clinician in the era of precision medicine
Nölting, S.; Ullrich, M.; Pietzsch, J.; Ziegler, C. G.; Eisenhofer, G.; et al. (7 authors)
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Cancers 11(2019), 1505
DOI: 10.3390/cancers11101505
ISSN: 2072-6694
Conventional CARs versus modular CARs
Feldmann, A.; Arndt, C.; Koristka, S.; Berndt, N.; Bergmann, R.; et al. (6 authors)
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Cancer Immunology, Immunotherapy 68(2019)10, 1713-1719
DOI: 10.1007/s00262-019-02399-5
A theranostic PSMA ligand for PET imaging and retargeting of T cells expressing the universal chimeric antigen receptor UniCAR
Arndt, C.; Feldmann, A.; Koristka, S.; Schäfer, M.; Bergmann, R.; et al. (19 authors)
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OncoImmunology 8(2019)9, 1659095
DOI: 10.1080/2162402X.2019.1659095
Biomaterials in repairing rat femoral defects: in vivo insights from small animal positron emission tomography/computed tomography (PET/CT) studies
Neuber, C.; Schulze, S.; Förster, Y.; Hofheinz, F.; Wodke, J.; et al. (11 authors)
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Clinical Hemorheology and Microcirculation 73(2019), 177-194
DOI: 10.3233/CH-199208
Theranostic CAR T cell targeting: A brief review
Arndt, C.; Bachmann, M.; Bergmann, R.; Berndt, N.; Feldmann, A.; et al. (6 authors)
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Journal of Labelled Compounds and Radiopharmaceuticals 62(2019)8, 533-540
DOI: 10.1002/jlcr.3727
Instant kit preparation of 68Ga-radiopharmaceuticals via the hybrid chelator DATA: clinical translation of [68Ga]Ga-DATA-TOC
Sinnes, J. P.; Nagel, J.; Waldron, B. P.; Maina, T.; Nock, B. A.; et al. (11 authors)
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EJNMMI Research 9(2019), 48
DOI: 10.1186/s13550-019-0516-7
Cytocompatible, Injectable, and Electroconductive Soft Adhesives with Hybrid Covalent/Noncovalent Dynamic Network
Xu, Y.; Patsis, P. A.; Hauser, S.; Voigt, D.; Rothe, R.; et al. (15 authors)
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Advanced Science 6(2019), 1802077
DOI: 10.1002/advs.201802077
T cells engrafted with a UniCAR 28/ζ outperform UniCAR BB/ζ-transduced T cells in the face of regulatory T cell-mediated immunosuppression
Kegler, A.; Koristka, S.; Bergmann, R.; Berndt, N.; Arndt, C.; et al. (10 authors)
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OncoImmunology 8(2019)9, e1621676
DOI: 10.1080/2162402X.2019.1621676
Nitric oxide-releasing selective estrogen receptor modulators (NO-SERMs): a bifunctional approach to improve the therapeutic index
Bechmann, N.; Knieß, T.; Pietzsch, J.
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Journal of Medicinal Chemistry 62(2019), 6525-6539
DOI: 10.1021/acs.jmedchem.9b00171
ISSN: 0022-2623
Targeting Cyclooxygenase-2 in Pheochromocytoma and Paraganglioma: Focus on Genetic Background
Ullrich, M.; Richter, S.; Seifert, V.; Hauser, S.; Calsina, B.; et al. (12 authors)
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Cancers 11(2019), 743
DOI: 10.3390/cancers11060743
ISSN: 2072-6694
Adjuvant drug-assisted bone healing: Part III – Further strategies for local and systemic modulation
Rothe, R.; Schulze, S.; Neuber, C.; Hauser, S.; Rammelt, S.; et al. (6 authors)
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Clinical Hemorheology and Microcirculation 73(2019), 439-488
DOI: 10.3233/CH-199104
ISSN: 1386-0291
Adjuvant drug-assisted bone healing: Part II – Modulation of angiogenesis
Rothe, R.; Schulze, S.; Neuber, C.; Hauser, S.; Rammelt, S.; et al. (6 authors)
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Clinical Hemorheology and Microcirculation 73(2019), 409-438
DOI: 10.3233/CH-199103
ISSN: 1386-0291
Adjuvant drug-assisted bone healing: Part I – Modulation of inflammation
Rothe, R.; Schulze, S.; Neuber, C.; Hauser, S.; Rammelt, S.; et al. (6 authors)
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Clinical Hemorheology and Microcirculation 73(2019), 381-408
DOI: 10.3233/CH-199102
ISSN: 1386-0291
Impact of Extrinsic and Intrinsic Hypoxia on Catecholamine Biosynthesis in Absence or Presence of Hif2α in Pheochromocytoma Cells
Bechmann, N.; Poser, I.; Seifert, V.; Greunke, C.; Ullrich, M.; et al. (13 authors)
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Cancers 11(2019), 594
DOI: 10.3390/cancers11050594
ISSN: 2072-6694
Carboranyl analogues of ketoprofen with cytostatic activity against human melanoma and colon cancer cell lines
Buzharevski, A.; Paskas, S.; Laube, M.; Lönnecke, P.; Neumann, W.; et al. (10 authors)
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ACS Omega 4(2019)5, 8824-8833
DOI: 10.1021/acsomega.9b00412
An oligo-His-tag of a targeting module does not influence its biodistribution and the retargeting capabilities of UniCAR T cells
Jureczek, J.; Bergmann, R.; Berndt, N.; Koristka, S.; Kegler, A.; et al. (10 authors)
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Scientific Reports 9(2019)1, 10547
DOI: 10.1038/s41598-019-47044-4
Limited importance of EphrinA1–ligand, Src kinase, and focal adhesion kinase in EphA2-mediated regulation of metastasis in Mel-Juso and A375 human melanoma cells
Neuber, C.; Herwig, N.; Pietzsch, J.; Belter, B.
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Journal of Cellular Biotechnology 5(2019)1, 11-26
DOI: 10.3233/JCB-189010
ISSN: 2352-3689
Regulation of A375 melanoma cell adhesion and migration by EphB4 and EphrinB2 –insights from co-culture experiments
Neuber, C.; Laube, M.; Mamat, C.; Belter, B.; Pietzsch, J.
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Journal of Cellular Biotechnology 5(2019)1, 27-42
DOI: 10.3233/JCB-189011
ISSN: 2352-3689
Radiochemical and radiopharmacological characterization of a 64Cu-labeled α-MSH analog conjugated with different chelators
Gao, F.; Sihver, W.; Bergmann, R.; Walther, M.; Stephan, H.; et al. (11 authors)
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Journal of Labelled Compounds and Radiopharmaceuticals 62(2019)8, 495-509
DOI: 10.1002/jlcr.3728
Fluorescent Mouse Pheochromocytoma Spheroids Expressing Hypoxia-Inducible Factor 2 alpha: Morphologic and Radiopharmacologic Characterization
Seifert, V.; Liers, J.; Kniess, T.; Richter, S.; Bechmann, N.; et al. (10 authors)
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Journal of Cellular Biotechnology 5(2019)2, 135-151
DOI: 10.3233/JCB-199005
ISSN: 2352-3689
Carboranyl Analogues of Celecoxib with Potent Cytostatic Activity against Human Melanoma and Colon Cancer Cell Lines
Buzharevski, A.; Paskas, S.; Sárosi, M. B.; Laube, M.; Lönnecke, P.; et al. (10 authors)
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ChemMedChem 14(2019)3, 315-321
DOI: 10.1002/cmdc.201800685
Fluorine-18 labeling of S100 proteins for small animal positron emission tomography
Laube, M.; Kniess, T.; Neuber, C.; Haase-Kohn, C.; Pietzsch, J.
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Methods in Molecular Biology 1929(2019), 461-485
DOI: 10.1007/978-1-4939-9030-6_29
ISSN: 1064-3745
Synthesis and preliminary radiopharmacological characterisation of an 11C-labelled azadipeptide nitrile as potential PET tracer for imaging of cysteine cathepsins
Laube, M.; Frizler, M.; Wodtke, R.; Neuber, C.; Belter, B.; et al. (10 authors)
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Journal of Labelled Compounds and Radiopharmaceuticals 62(2019)8, 448-459
DOI: 10.1002/jlcr.3729
Synthesis, 18F-labelling and radiopharmacological characterisation of the C-terminal 30mer of Clostridium perfringens enterotoxin as a potential claudin-targeting peptide
Löser, R.; Bader, M.; Kuchar, M.; Wodtke, R.; Lenk, J.; et al. (12 authors)
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Amino Acids 51(2019)2, 219-244
Online First (2018) DOI: 10.1007/s00726-018-2657-9
One-pot Cascade Synthesis of Pyrazole-based Isosteres of Valdecoxib by a [3+2] Cycloaddition/[1,5] Sigmatropic Rearrangement Sequence and Evaluation of their COX Inhibitory Activity
Roscales, S.; Bechmann, N.; Pietzsch, J.; Kniess, T.
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Heterocycles 98(2019)3, 416-428
DOI: 10.3987/COM-19-14048
Anti-CAR engineered T cells for epitope-based elimination of autologous CAR T cells
Koristka, S.; Ziller-Walter, P.; Bergmann, R.; Arndt, C.; Feldmann, A.; et al. (11 authors)
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Cancer Immunology, Immunotherapy (2019), 1401-1415
DOI: 10.1007/s00262-019-02376-y
Access to 18F-labelled isoxazoles by Ruthenium-promoted 1,3-dipolar cycloaddition of 4-[18F]fluoro-N-hydroxybenzimidoyl chloride with alkynes.
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Journal of Labelled Compounds and Radiopharmaceuticals 62(2019), 393-403
DOI: 10.1002/jlcr.3708
2018
Evaluation of Brain Nuclear Medicine Imaging Tracers in a Murine Model of Sepsis-Associated Encephalopathy
Szöllősi, D.; Hegedűs, N.; Veres, D. S.; Futó, I.; Horváth, I.; et al. (15 authors)
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Molecular Imaging and Biology 20(2018), 952-962
DOI: 10.1007/s11307-018-1201-3
Multimodal PET/MRI Imaging Results Enable Monitoring the Side Effects of Radiation Therapy.
Kovács, N.; Szigeti, K.; Hegedűs, N.; Horváth, I.; Veres, D. S.; et al. (8 authors)
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Contrast Media & Molecular Imaging (2018), 5906471
DOI: 10.1155/2018/5906471
Diverse Effects of Phospholipase A2 Receptor Expression on LNCaP and PC-3 Prostate Cancer Cell Growth in vitro and in vivo
Friedemann, M.; Nacke, B.; Hagelgans, A.; Jandeck, C.; Bechmann, N.; et al. (11 authors)
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Oncotarget 9(2018), 35983-35996
DOI: 10.18632/oncotarget.26316
Improved Conjugation, 64-Cu Radiolabeling, in Vivo Stability, and Imaging Using Nonprotected Bifunctional Macrocyclic Ligands: Bis(Phosphinate) Cyclam (BPC) Chelators
David, T.; Hlinová, V.; Kubíček, V.; Bergmann, R.; Striese, F.; et al. (12 authors)
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Journal of Medicinal Chemistry 61(2018), 8774-8796
DOI: 10.1021/acs.jmedchem.8b00932
Synthesis, characterization and initial biological evaluation of [⁹⁹ᵐTc]Tc-tricarbonyl labeled DPA-α-MSH peptide derivatives for potential melanoma imaging
Gao, F.; Sihver, W.; Bergmann, R.; Belter, B.; Bolzati, C.; et al. (9 authors)
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ChemMedChem 13(2018)11, 1146-1158
DOI: 10.1002/cmdc.201800110
Exploring pitfalls of 64Cu‑labeled EGFR‑targeting peptide GE11 as a potential PET tracer
Striese, F.; Sihver, W.; Gao, F.; Bergmann, R.; Walther, M.; et al. (8 authors)
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Amino Acids 50(2018)10, 1415-1431
DOI: 10.1007/s00726-018-2616-5
Development of a novel target module redirecting UniCAR T cells to Sialyl Tn-expressing tumor cells
Loureiro, L.; Feldmann, A.; Bergmann, R.; Koristka, S.; Berndt, N.; et al. (10 authors)
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Blood Cancer Journal 8(2018), 81
DOI: 10.1038/s41408-018-0113-4
Strain-specific metastatic phenotypes in pheochromocytoma allograft mice
Ullrich, M.; Liers, J.; Peitzsch, M.; Feldmann, A.; Bergmann, R.; et al. (12 authors)
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Endocrine-Related Cancer 25(2018)12, 993-1004
DOI: 10.1530/ERC-18-0136
From mono- to bivalent: improving theranostic properties of target modules for redirection of UniCAR T cells against EGFR-expressing tumor cells in vitro and in vivo
Albert, S.; Arndt, C.; Koristka, S.; Berndt, N.; Bergmann, R.; et al. (10 authors)
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Oncotarget 9(2018)39, 25597-25616
DOI: 10.18632/oncotarget.25390
Nε-Acryloyllysine piperazides as irreversible inhibitors of transglutaminase 2 – synthesis, structure-activity relationships and pharmacokinetic profiling
Wodtke, R.; Hauser, C.; Ruiz-Gómez, G.; Jäckel, E.; Bauer, D.; et al. (16 authors)
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Journal of Medicinal Chemistry 61(2018)10, 4528-4560
DOI: 10.1021/acs.jmedchem.8b00286
Biodistribution studies of ultrasmall silicon nanoparticles and carbon dots in experimental rats and tumor mice
Licciardello, N.; Hunoldt, S.; Bergmann, R.; Singh, G.; Mamat, C.; et al. (11 authors)
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Nanoscale 10(2018), 9880-9891
DOI: 10.1039/C8NR01063C
Overexpression of receptor tyrosine kinase EphB4 triggers tumor growth and hypoxia in A375 melanoma xenografts: insights from multitracer small animal imaging experiments
Neuber, C.; Belter, B.; Meister, S.; Hofheinz, F.; Bergmann, R.; et al. (7 authors)
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Molecules 23(2018), 444
DOI: 10.3390/molecules23020444
Bridging from Brain to Tumor imaging: (S)- and (R)-[18F]Fluspidine for investigation of Sigma-1 Receptors in Tumor-bearing Mice
Kranz, M.; Bergmann, R.; Kniess, T.; Belter, B.; Neuber, C.; et al. (14 authors)
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Molecules 23(2018)3, 702
DOI: 10.3390/molecules23030702
Causative treatment of acid aspiration induced acute lung injury – recent trends from animal experiments and critical perspective
Gramatté, J.; Pietzsch, J.; Bergmann, R.; Richter, T.
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Clinical Hemorheology and Microcirculation 69(2018), 187-195
DOI: 10.3233/CH-189113
ISSN: 1386-0291
Engrafting human regulatory T cells with a flexible modular chimeric antigen receptor technology
Koristka, S.; Kegler, A.; Bergmann, R.; Arndt, C.; Feldmann, A.; et al. (17 authors)
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Journal of Autoimmunity 90(2018), 116-131
DOI: 10.1016/j.jaut.2018.02.006
Evaluation of fluorine-18-labelled alpha1(I)-N-telopeptide analogues as substrate-based radiotracers for PET imaging of melanoma-associated lysyl oxidase
Kuchar, M.; Neuber, C.; Belter, B.; Bergmann, R.; Lenk, J.; et al. (10 authors)
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Frontiers in Chemistry 6(2018), 121
DOI: 10.3389/fchem.2018.00121
Novel Valdecoxib Derivates by Ruthenium-catalyzed 1,3-Dipolar Cycloaddition of Nitrile Oxides with Alkynes - Synthesis and COX-2 Inhibition Affinity.
Roscales, S.; Bechmann, N.; Weiss, D. H.; Köckerling, M.; Pietzsch, J.; et al. (6 authors)
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MedChemComm 9(2018), 534-544
DOI: 10.1039/c7md00575j
2017
An orthotopic xenograft model for high-risk non-muscle invasive bladder cancer in mice: influence of mouse strain, tumor cell count, dwell time and bladder pretreatment
Huebner, D.; Rieger, C.; Bergmann, R.; Ullrich, M.; Meister, S.; et al. (13 authors)
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BMC Cancer 17(2017)1, 790
DOI: 10.1186/s12885-017-3778-3
Novel Radiolabeled Bisphosphonates for PET Diagnosis and Endoradiotherapy of Bone Metastases
Pfannkuchen, N.; Meckel, M.; Bergmann, R.; Bachmann, M.; Bal, C.; et al. (9 authors)
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Pharmaceuticals 10(2017), 45
DOI: 10.3390/ph10020045
Biological characterization of novel nitroimidazole-peptide conjugates in vitro and in vivo.
Bergmann, R.; Splith, K.; Pietzsch, J.; Bachmann, M.; Neundorf, I.
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Journal of Peptide Science 23(2017), 597-609
DOI: 10.1002/psc.2995
Characterization of a switchable chimeric antigen receptor platform in a pre-clinical solid tumor model
Bejestani, E. P.; Cartellieri, M.; Bergmann, R.; Ehninger, A.; Loff, S.; et al. (17 authors)
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OncoImmunology 6(2017)10, 1342909
DOI: 10.1080/2162402X.2017.1342909
Retargeting of UniCAR T cells with an in vivo synthesized target module directed against CD19 positive tumor cells
Bachmann, D.; Aliperta, R.; Bergmann, R.; Feldmann, A.; Koristka, S.; et al. (19 authors)
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Oncotarget 9(2017), 7487-7500
DOI: 10.18632/oncotarget.23556
Development of novel target modules for retargeting of UniCAR T cells to GD2 positive tumor cells
Mitwasi, N.; Feldmann, A.; Bergmann, R.; Berndt, N.; Arndt, C.; et al. (17 authors)
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Oncotarget 8(2017), 108584-108603
DOI: 10.18632/oncotarget.21017
99mTechnetium-based Small Molecule Radiopharmaceuticals and Radiotracers Targeting Inflammation and Infection
Kniess, T.; Laube, M.; Wüst, F.; Pietzsch, J.
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Dalton Transactions 46(2017), 14435-14451
DOI: 10.1039/c7dt01735a
Preparation of a novel radiotracer targeting the EphB4 receptor via radiofluorination using spiro azetidinium salts as precursor
Wiemer, J.; Steinbach, J.; Pietzsch, J.; Mamat, C.
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Journal of Labelled Compounds and Radiopharmaceuticals 60(2017), 489-498
DOI: 10.1002/jlcr.3526
Surface charge and particle size determine the metabolic fate of dendritic polyglycerols
Pant, K.; Pufe, J.; Zarschler, K.; Bergmann, R.; Steinbach, J.; et al. (9 authors)
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Nanoscale 9(2017), 8723-8739
DOI: 10.1039/C7NR01702B
A novel nanobody-based target module for retargeting of T lymphocytes to EGFR-expressing cancer cells via the modular UniCAR platform
Albert, S.; Arndt, C.; Feldmann, A.; Bergmann, R.; Bachmann, D.; et al. (18 authors)
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OncoImmunology 6(2017)4, e1287246
DOI: 10.1080/2162402X.2017.1287246
ISSN: 2162-402X
A novel tumor pretargeting system based on complementary L-configured oligonucleotides
Schubert, M.; Bergmann, R.; Förster, C.; Sihver, W.; Vonhoff, S.; et al. (12 authors)
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Bioconjugate Chemistry 28(2017)4, 1176-1188
DOI: 10.1021/acs.bioconjchem.7b00045
Distribution and kinetics of the Kv1.3-blocking peptide HsTX1[R14A] in experimental rats
Bergmann, R.; Kubeil, M.; Zarschler, K.; Chhabra, S.; Tajhya, R. B.; et al. (10 authors)
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Scientific Reports 7(2017), 3756
DOI: 10.1038/s41598-017-03998-x
In vivo examination of an injectable hydrogel system crosslinked by peptide-oligosaccharide interaction in immunocompetent nude mice
Tondera, C.; Wieduwild, R.; Röder, E.; Werner, C.; Zhang, Y.; et al. (6 authors)
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Advanced Functional Materials 27(2017)15, 1605189
DOI: 10.1002/adfm.201605189
Development of Fluorinated Non-Peptidic Ghrelin Receptor Ligands for Potential Use in Molecular Imaging
Moldovan, R.-P.; Els-Heindl, S.; Worm, D. J.; Kniess, T.; Kluge, M.; et al. (9 authors)
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International Journal of Molecular Sciences 18(2017)4, 768
DOI: 10.3390/ijms18040768
Retargeting of T lymphocytes to PSCA- or PSMA positive prostate cancer cells using the novel modular chimeric antigen receptor platform technology “UniCAR”
Feldmann, A.; Arndt, C.; Bergmann, R.; Loff, S.; Cartellieri, M.; et al. (20 authors)
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Oncotarget 8(2017)19, 31368-31385
DOI: 10.18632/oncotarget.15572
The Why and How of Amino Acid Analytics in Cancer Diagnostics and Therapy
Manig, F.; Kuhne, K.; von Neubeck, C.; Schwarzenbolz, U.; Yu, Z.; et al. (8 authors)
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Journal of Biotechnology 242(2017), 30-54
DOI: 10.1016/j.jbiotec.2016.12.001
Human endothelial cell models in biomaterial research
Hauser, S.; Jung, F.; Pietzsch, J.
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Trends in Biotechnology 35(2017)3, 265-277
DOI: 10.1016/j.tibtech.2016.09.007
Hydrous 18F-fluoroethylation – leaving off the azeotropic drying
Kniess, T.; Laube, M.; Steinbach, J.
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Applied Radiation and Isotopes 127(2017), 260-268
DOI: 10.1016/j.apradiso.2017.06.010
ISSN: 0969-8043
Cryogel-Supported Stem Cell Factory for Customized Sustained Release of Bispecific Antibodies for Cancer Immunotherapy
Aliperta, R.; Welzel, P. B.; Bergmann, R.; Freudenberg, R.; Berndt, N.; et al. (17 authors)
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Scientific Reports 7(2017), 42855
DOI: 10.1038/srep42855
Insights into binding of S100 proteins to scavenger receptors: class B scavenger receptor CD36 binds S100A12 with high affinity
Tondera, C.; Laube, M.; Pietzsch, J.
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Amino Acids 49(2017), 183-191
Online First (2016) DOI: 10.1007/s00726-016-2349-2
2016
Radiomics-based differentiation of lung disease models generated by polluted air based on X-ray computed tomography data
Szigeti, K.; Szabó, T.; Korom, C.; Ilona, C.; Horváth, I.; et al. (12 authors)
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BMC Medical Imaging 16(2016), 14
DOI: 10.1186/s12880-016-0118-z
Development of a F-18-labeled Diaryl-Substituted Dihydropyrrolo[3,2,1-hi]indole as Potential Probe for Functional Imaging of Cyclooxygenase-2 with PET
Gassner, C.; Neuber, C.; Laube, M.; Bergmann, R.; Kniess, T.; et al. (6 authors)
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ChemistrySelect 1(2016), 5812-5820
DOI: 10.1002/slct.201601618
ISSN: 2365-6549
Gelatin-based hydrogel degradation and tissue interaction in vivo: insights from multimodal preclinical imaging in immunocompetent nude mice
Tondera, C.; Ullm, S.; Krüger-Genge, A.; Jung, F.; Neffe, A. T.; et al. (10 authors)
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Theranostics 6(2016)12, 2114-2128
DOI: 10.7150/thno.16614
Zwitterionic polymer-coated ultrasmall superparamagnetic iron oxide nanoparticles with low protein interaction and high biocompatibility
Pombo-García, K.; Weiss, S.; Zarschler, K.; Ang, C.-S.; Hübner, R.; et al. (12 authors)
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ChemNanoMat 2(2016)10, 959-971
DOI: 10.1002/cnma.201600233
Extracellular S100A4 affects endothelial cell integrity and stimulates transmigratory behavior of human A375 melanoma cells
Herwig, N.; Belter, B.; Pietzsch, J.
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Biochemical and Biophysical Research Communications 477(2016)4, 963-969
DOI: 10.1016/j.bbrc.2016.07.009
Synthesis and kinetic characterisation of water-soluble fluorogenic acyl donors for transglutaminase 2
Wodtke, R.; Schramm, G.; Pietzsch, J.; Pietsch, M.; Löser, R.
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ChemBioChem 17(2016), 1263-1281
DOI: 10.1002/cbic.201600048
Multimodal Somatostatin Receptor Theranostics Using [64Cu]Cu-/[177Lu]Lu-DOTA-(Tyr3)octreotate and AN-238 in a Mouse Pheochromocytoma Model.
Ullrich, M.; Bergmann, R.; Peitzsch, M.; Zenker, E.; Cartellieri, M.; et al. (13 authors)
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Theranostics 6(2016)5, 650-665
DOI: 10.7150/thno.14479
Development of antioxidant COX-2 inhibitors as radioprotective agents for radiation therapy – a hypothesis-driven review
Laube, M.; Kniess, T.; Pietzsch, J.
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Antioxidants 5(2016)2, 14
DOI: 10.3390/antiox5020014
5-Chloro-1-phenylpentan-1-one
Bechmann, N.; Kniess, T.; Pietzsch, J.; König, J.; Köckerling, M.
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IUCrData 1(2016), 160055
DOI: 10.1107/S2414314616000559
ISSN: 2414-3146
177Lu-labelled macrocyclic bisphosphonates for targeting bone metastasis in cancer treatment
Bergmann, R.; Meckel, M.; Kubicek, V.; Pietzsch, J.; Steinbach, J.; et al. (7 authors)
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EJNMMI Research 6(2016)1, 5
DOI: 10.1186/s13550-016-0161-3
Radiopharmacological characterization of 64Cu-labeled α-MSH analogs for potential use in imaging of malignant melanoma
Gao, F.; Sihver, W.; Jurischka, C.; Bergmann, R.; Haase-Kohn, C.; et al. (12 authors)
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Amino Acids 48(2016)3, 833-847
Online First (2015) DOI: 10.1007/s00726-015-2131-x
Interaction of extracellular S100A4 with RAGE prompts prometastatic activation of A375 melanoma cells
Herwig, N.; Belter, B.; Wolf, S.; Haase-Kohn, C.; Pietzsch, J.
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Journal of Cellular and Molecular Medicine 20(2016)5, 825-835
DOI: 10.1111/jcmm.12808
2015
Protective effects of 2,3-diaryl-substituted indole-based cyclooxygenase-2 inhibitors on oxidative modification of human low density lipoproteins in vitro
Pietzsch, J.; Laube, M.; Bechmann, N.; Pietzsch, F.-J.; Kniess, T.
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Clinical Hemorheology and Microcirculation 61(2015)4, 615-632
DOI: 10.3233/CH-141923
ISSN: 1386-0291
Controlled immobilization of His-tagged proteins for protein-ligand interaction experiments using Ni2+-NTA layer on glass surfaces
Cherkouk, C.; Rebohle, L.; Lenk, J.; Keller, A.; Ou, X.; et al. (10 authors)
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Clinical Hemorheology and Microcirculation 61(2015), 523
DOI: 10.3233/CH-151950
Influence of irradiation on release of endothelial microparticles (EMP) in vitro
Neuber, C.; Pufe, J.; Pietzsch, J.
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Clinical Hemorheology and Microcirculation 61(2015)2, 291-299
DOI: 10.3233/CH-151987
ISSN: 1386-0291
18F-Labeled 1,4-Dioxa-8-azaspiro[4.5]decane Derivative: Synthesis and Biological Evaluation of a σ1 Receptor Radioligand with Low Lipophilicity as Potent Tumor Imaging Agent
Xie, F.; Bergmann, R.; Kniess, T.; Deuther-Conrad, W.; Mamat, C.; et al. (11 authors)
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Journal of Medicinal Chemistry 58(2015), 5395-5407
DOI: 10.1021/acs.jmedchem.5b00593
ISSN: 0022-2623
2-[18F]Fluoroethyl tosylate - a versatile tool for building 18F-based radiotracers for positron emission tomography
Knieß, T.; Laube, M.; Brust, P.; Steinbach, J.
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MedChemComm 6(2015), 1714-1754
DOI: 10.1039/c5md00303b
Novel (pyrazolyl)benzenesulfonamides with a nitric oxide-releasing moiety as selective cyclooxygenase-2 inhibitors
Bechmann, N.; Kniess, T.; Köckerling, M.; Pigorsch, A.; Steinbach, J.; et al. (6 authors)
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