Publications of Institute of Radiopharmaceutical Cancer Research
409 Publications2014
Bispidine dioxotetraaza macrocycles: a new class of bispidines for 64Cu PET imaging
Comba, P.; Kubeil, M.; Pietzsch, J.; Rudolf, H.; Stephan, H.; et al. (6 authors)
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Inorganic Chemistry 53(2014), 6698-6707
DOI: 10.1021/ic500476u
Radiofluorination and first radiopharmacological characterization of a SWLAY peptide-based ligand targeting EphA2
Pretze, M.; Mosch, B.; Bergmann, R.; Steinbach, J.; Pietzsch, J.; et al. (6 authors)
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Journal of Labelled Compounds and Radiopharmaceuticals 57(2014), 660-665
DOI: 10.1002/jlcr.3237
Effect of [18F]FMISO stratified dose-escalation on local control in FaDu hSCC in nude mice
Schütze, C.; Bergmann, R.; Brüchner, K.; Mosch, B.; Yaromira, A.; et al. (13 authors)
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Radiotherapy and Oncology 111(2014), 81-87
DOI: 10.1016/j.radonc.2014.02.005
ISSN: 1879-0887
Metastatic potential of B16-F10 melanoma cells is enhanced by extracellular S100A4 derived from RAW264.7 macrophages
Haase-Kohn, C.; Wolf, S.; Herwig, N.; Mosch, B.; Pietzsch, J.
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Biochemical and Biophysical Research Communications 446(2014), 143-148
DOI: 10.1016/j.bbrc.2014.02.126
Influence of different chelators on the radiochemical properties of a 68-Gallium labelled bombesin analogue.
Asti, M.; Iori, M.; Capponi, P. C.; Atti, G.; Rubagotti, S.; et al. (11 authors)
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Nuclear Medicine and Biology 41(2014), 24-35
DOI: 10.1016/j.nucmedbio.2013.08.010
Radiolabeled anti-EGFR-antibody improves local tumor control after external beam radiotherapy and offers theragnostic potential
Koi, L.; Bergmann, R.; Brüchner, K.; Pietzsch, J.; Pietzsch, H.-J.; et al. (9 authors)
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Radiotherapy and Oncology 110(2014), 362-369
DOI: 10.1016/j.radonc.2013.12.001
Radiolabeled cetuximab conjugates for EGFR targeted cancer diagnostics and therapy
Sihver, W.; Pietzsch, J.; Krause, M.; Baumann, M.; Steinbach, J.; et al. (6 authors)
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Pharmaceuticals 7(2014)3, 311-338
DOI: 10.3390/ph7030311
2013
Pulmonary Blood Flow Increases in Damaged Regions Directly after Acid Aspiration in Rats
Richter, T.; Bergmann, R.; Knels, L.; Hofheinz, F.; Kasper, M.; et al. (9 authors)
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Anesthesiology 119(2013), 890-900
DOI: 10.1097/ALN.0b013e3182a17e5b
ISSN: 0003-3022
Synthesis and radiopharmacological evaluation of 64Cu-labeled bombesin analogs featuring a bis(2-pyridylmethyl) 1,4,7-triazacyclononane chelator
Bergmann, R.; Ruffani, A.; Graham, B.; Spiccia, L.; Steinbach, J.; et al. (7 authors)
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European Journal of Medicinal Chemistry 70(2013), 434-446
DOI: 10.1016/j.ejmech.2013.10.013
Tissue transglutaminase: an emerging target for therapy and imaging
Pietsch, M.; Wodtke, R.; Pietzsch, J.; Löser, R.
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Bioorganic & Medicinal Chemistry Letters 23(2013)24, 6528-6543
DOI: 10.1016/j.bmcl.2013.09.060
In vivo comparison of DOTA based 68Ga-labelled bisphosphonates for bone imaging in non-tumour models
Meckel, M.; Fellner, M.; Thieme, N.; Bergmann, R.; Kubicek, V.; et al. (6 authors)
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Nuclear Medicine and Biology 40(2013), 823-830
DOI: 10.1016/j.nucmedbio.2013.04.012
Synthesis and radiopharmacological evaluation of a high-affinity and metabolically stabilized 18F-labeled bombesin analogue for molecular imaging of gastrin-releasing peptide receptor-expressing prostate cancer
Richter, S.; Wuest, M.; Krieger, S. S.; Rogers, B. E.; Friebe, M.; et al. (7 authors)
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Nuclear Medicine and Biology 40(2013), 1025-1034
DOI: 10.1016/j.nucmedbio.2013.07.005
Radiosynthesis and in vivo Evaluation of a 18F-Labelled Styryl-Benzoxazole Derivative for ß-Amyloid Targeting
Ribeiro Morais, G.; Kniess, T.; Bergmann, R.; Gano, L.; Abrunhosa, A.; et al. (7 authors)
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Applied Radiation and Isotopes 82(2013), 100-104
DOI: 10.1016/j.apradiso.2013.07.003
Optimization of Pentadentate Bispidines as Bifunctional Chelators for 64Cu Positron Emission Tomography (PET)
Comba, P.; Hunoldt, S.; Morgen, M.; Pietzsch, J.; Stephan, H.; et al. (6 authors)
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Inorganic Chemistry 52(2013), 8131-8143
DOI: 10.1021/ic4008685
An Efficient Bioorthogonal Strategy Using CuAAC Click Chemistry for Radiofluorinations of SNEW Peptides and the Role of Copper Depletion
Pretze, M.; Kuchar, M.; Bergmann, R.; Steinbach, J.; Pietzsch, J.; et al. (6 authors)
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ChemMedChem 8(2013), 935-945
DOI: 10.1002/cmdc.201300053
Synthesis and radiopharmacological characterisation of a fluorine-18 labelled azadipeptide nitrile as potential PET Tracer for in vivo imaging of cysteine cathepsins
Löser, R.; Bergmann, R.; Frizler, M.; Mosch, B.; Dombrowski, L.; et al. (9 authors)
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ChemMedChem 8(2013), 1330-1344
DOI: 10.1002/cmdc.201300135
Recent trends in malignant melanoma biomarker research
Pietzsch, J.; Tandler, N.; Mosch, B.
- Clinical Laboratory International 37(2013), 6-8
Anti-tumor effects of peptide analogues targeting neuropeptide hormone receptors on mouse pheochromocytoma cells
Ziegler, C. G.; Eisenhofer, G.; Schally, A. V.; Gebauer, L.; Gondek, K.; et al. (11 authors)
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Molecular and Cellular Endocrinology 371(2013), 189-194
DOI: 10.1016/j.mce.2012.12.011
ISSN: 0303-7207
Radiolabeled COX-2 inhibitors for non-invasive visualization of COX-2 expression and activity - a critical update
Laube, M.; Kniess, T.; Pietzsch, J.
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Molecules 18(2013), 6311-6355
DOI: 10.3390/molecules18066311
Ga-68- and Cu-64-Labeled NOTA-Albumin Conjugates for PET Sentinel Lymph Node Imaging
Schiller, E.; Bergmann, R.; Wunderlich, G.; Andreeff, M.; Jacob, A.; et al. (6 authors)
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ISRN Molecular Imaging (2013), 386976
DOI: 10.1155/2013/386976
Experimental hypoxia does not influence gene expression and protein synthesis of Eph receptors and ephrin ligands in human melanoma cells in vitro.
Reissenweber, B.; Mosch, B.; Pietzsch, J.
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Melanoma Research 23(2013), 85-95
DOI: 10.1097/CMR.0b013e32835e58f3
Investigations into the synthesis, radiofluorination and conjugation of a new [18F]fluorocyclobutyl prosthetic group and its in vitro stability using a tyrosine model system
Franck, D.; Kniess, T.; Steinbach, J.; Zitzmann-Kolbe, S.; Friebe, M.; et al. (7 authors)
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Bioorganic & Medicinal Chemistry 21(2013), 643-652
DOI: 10.1016/j.bmc.2012.11.049
Visualization of cyclooxygenase-2 using a 2,3-diarylsubstituted indole-based inhibitor and confocal laser induced cryofluorescence microscopy at 20 K in melanoma cells in vitro
Tondera, C.; Laube, M.; Wimmer, C.; Kniess, T.; Mosch, B.; et al. (7 authors)
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Biochemical and Biophysical Research Communications 430(2013), 301-306
Online First (2012) DOI: 10.1016/j.bbrc.2012.10.133
Copper(II) chemistry of the functionalized macrocycle cyclam tetrapropionic acid
Comba, P.; Emmerling, F.; Jakob, M.; Kraus, W.; Kubeil, M.; et al. (8 authors)
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Dalton Transactions 42(2013), 6142-6148
Online First (2012) DOI: 10.1039/C2DT32356G
2-Carbaborane-3-phenyl-1H-indoles—Synthesis via McMurry Reaction and Cyclooxygenase (COX) Inhibition Activity
Laube, M.; Neumann, W.; Scholz, M.; Lönnecke, P.; Crews, B.; et al. (9 authors)
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ChemMedChem 8(2013)2, 329-335
DOI: 10.1002/cmdc.201200455
2012
Cerebral blood flow quantification in the rat: a direct comparison of arterial spin labeling MRI with radioactive microsphere PET
Bos, A.; Bergmann, R.; Strobel, K.; Hofheinz, F.; Steinbach, J.; et al. (6 authors)
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EJNMMI Research 2(2012)47
DOI: 10.1186/2191-219X-2-47
ISSN: 2191-219X
Protein and non-protein biomarkers in melanoma: a critical update.
Tandler, N.; Mosch, B.; Pietzsch, J.
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Amino Acids 6(2012), 2203-2230
DOI: 10.1007/s00726-012-1409-5
Synthesis, in silico, in vitro, and in vivo investigation of 5-[11C]methoxy-substituted sunitinib, a tyrosine kinase inhibitor of VEGFR-2
Caballero, J.; Muñoz, C.; Alzate-Morales, J. H.; Cunha, S.; Gano, L.; et al. (8 authors)
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European Journal of Medicinal Chemistry 58(2012), 272-280
DOI: 10.1016/j.ejmech.2012.10.020
18F-Labeled phosphopeptide-cell-penetrating peptide dimers with enhanced cell uptake properties in human cancer cells
Richter, S.; Bouvet, V.; Wuest, M.; Bergmann, R.; Steinbach, J.; et al. (8 authors)
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Nuclear Medicine and Biology 39(2012)8, 1202-1212
DOI: 10.1016/j.nucmedbio.2012.06.003
Synthesis and cytotoxicity of pyridine and quinoline oxorhenium(V) complexes with tridentate (NS2, S-3)/monodentate (s) coordination
Segal, I.; Zablotskaya, A.; Kniess, T.; Shestakova, I.
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Chemistry of Heterocyclic Compounds 48(2012), 296-300
DOI: 10.1007/s10593-012-0989-z
ISSN: 0009-3122
18F-labelled CCR1-receptor antagonist is not suitable for imaging of Alzheimer's disease
Beuthien-Baumann, B.; Holthoff, V.; Mäding, P.; Bergmann, R.; Pawelke, B.; et al. (9 authors)
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Nuklearmedizin 51(2012), 239-243
DOI: 10.3413/Nukmed-0457-12-01
ISSN: 0029-5566
Fluorine-18-Radiolabeling and Radiopharmacological Characterization of a Benzodioxolylpyrimidine as a Radiotracer Targeting the Receptor Tyrosine Kinase EphB4
Mamat, C.; Mosch, B.; Neuber, C.; Köckerling, M.; Bergmann, R.; et al. (6 authors)
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ChemMedChem 7(2012)11, 1991-2003
DOI: 10.1002/cmdc.201200264
Novel 7α-alkoxy-17α-(4’-halophenylethynyl)estradiols as potential SPECT/PET imaging agents for estrogen receptor expressing tumors: synthesis and binding affinity evaluation
Neto, C.; Oliveira, M. C.; Gano Fernanda Marques, M. L.; Yasuda, T.; Thiemann, T.; et al. (7 authors)
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Steroids 77(2012), 1123-1132
DOI: 10.1016/j.steroids.2012.05.004
Design, Evaluation, and Comparison of Ghrelin Receptor Agonists and Inverse Agonists as Suitable Radiotracers for PET Imaging
Chollet, C.; Bergmann, R.; Pietzsch, J.; Beck-Sickinger, A. G.
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Bioconjugate Chemistry 23(2012), 771-784
DOI: 10.1021/bc2005889
Irradiation affects cellular properties and Eph receptor expression in human melanoma cells
Mosch, B.; Pietzsch, D.; Pietzsch, J.
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Cell Adhesion & Migration 6(2012)2, 113-125
DOI: 10.4161/cam.20655
ISSN: 1933-6918
Radioiodinated sunitinib as a potential radiotracer for imaging angiogenesis - radiosynthesis and first radiopharmacological evaluation of 5-[125I]Iodo-sunitinib
Kuchar, M.; Oliveira, M. C.; Gano, L.; Santos, I.; Knieß, T.
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Bioorganic & Medicinal Chemistry Letters 22(2012), 2850-2855
DOI: 10.1016/j.bmcl.2012.02.068
Radiohalogenated 4-anilinoquinazoline-based EGFR-TK inhibitors as potential cancer imaging agents
Neto, C.; Fernandes, C.; Oliveira, M. C.; Gano, L.; Mendes, F.; et al. (7 authors)
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Nuclear Medicine and Biology 39(2012), 247-260
DOI: 10.1016/j.nucmedbio.2011.09.001
Study of differences in the VEGFR2 inhibitory activities between semaxanib and SU5205 using 3D-QSAR, docking, and molecular dynamics simulations
Munoza, C.; Adasmea, F.; Alzate-Morales, J. H.; Vergara-Jaquea, A.; Kniess, T.; et al. (6 authors)
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Journal of Molecular Graphics and Modelling 32(2012), 39-48
DOI: 10.1016/j.jmgm.2011.10.005
Radiolabeled small molecule inhibitors of VEGFR – recent advances
Kniess, T.
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Current Pharmaceutical Design 18(2012), 2867-2874
DOI: 10.2174/138161212800672796
ISSN: 1873-4286
Specific targeting of hypoxic tumor tissue with nitroimidazole-peptide conjugates
Splith, K.; Bergmann, R.; Pietzsch, J.; Neundorf, I.
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ChemMedChem 7(2012), 57-61
DOI: 10.1002/cmdc.201100401
Site-selective radiolabeling of peptides by 18F-fluorobenzoylation with [18F]SFB in solution and on solid phase - a comparative study
Kuchar, M.; Pretze, M.; Knieß, T.; Steinbach, J.; Pietzsch, J.; et al. (6 authors)
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Amino Acids 43(2012), 1431-1443
DOI: 10.1007/s00726-012-1216-z
Radiosynthesis of a 18F-labeled 2,3-diarylsubstituted indole via McMurry coupling for functional characterization of cyclooxygenase-2 (COX-2) in vitro and in vivo
Kniess, T.; Laube, M.; Bergmann, R.; Graf, F.; Steinbach, J.; et al. (7 authors)
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Bioorganic & Medicinal Chemistry 20(2012), 3410-3421
DOI: 10.1016/j.bmc.2012.04.022
2011
Synthesis of an 18F-labeled cyclin-dependent kinase-2 inhibitor
Svensson, F.; Kniess, T.; Bergmann, R.; Pietzsch, J.; Wuest, F.
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Journal of Labelled Compounds and Radiopharmaceuticals 54(2011), 769-774
DOI: 10.1002/jlcr.1922
S100A2 in cancerogenesis: a friend or a foe?
Wolf, S.; Haase-Kohn, C.; Pietzsch, J.
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Amino Acids 41(2011), 849-861
DOI: 10.1007/s00726-010-0623-2
S100 proteins in health and disease
Pietzsch, J.
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Amino Acids 41(2011), 755-760
DOI: 10.1007/s00726-010-0816-8
Influence of storage on the position of the germinal disc in the fertilized unincubated chicken egg
Burkhardt, A.; Meister, S.; Bergmann, R.; Koch, E.
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Poultry Science 90(2011), 2169-2173
DOI: 10.3382/ps.2010-01179
ISSN: 0032-5791
Copper-mediated cross-linking of S100A4, but not of S100A2, results in proinflammatory effects in melanoma cells
Haase-Kohn, C.; Wolf, S.; Lenk, J.; Pietzsch, J.
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Biochemical and Biophysical Research Communications 413(2011), 494-498
DOI: 10.1016/j.bbrc.2011.08.132
Phosphopeptides with improved cellular uptake properties as ligands for the polo-box domain of polo-like kinase 1
Richter, S.; Neundorf, I.; Loebner, K.; Gräber, M.; Berg, T.; et al. (9 authors)
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Bioorganic & Medicinal Chemistry Letters 21(2011), 4686-4689
DOI: 10.1016/j.bmcl.2011.06.103
Impact of functionalized coligands on the pharmacokinetics of 99mTc(III) ‘4+1’ mixed-ligand complexes conjugated to bombesin
Künstler, J.-U.; Bergmann, R.; Gniazdowska, E.; Kozminski, P.; Walther, M.; et al. (6 authors)
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Journal of Inorganic Biochemistry 105(2011), 1383-1390
DOI: 10.1016/j.jinorgbio.2011.07.002
Radiolabeling of phosphatidylserine-binding peptides with prosthetic groups N-[6-(4-[18F]fluorobenzylidene)aminooxyhexyl]maleimide ([18F]FBAM) and N-succinimidyl-4-[18F]fluorobenzoate ([18F]SFB)
Kapty, J.; Kniess, T.; Wuest, F.; Mercer, J. R.
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Applied Radiation and Isotopes 69(2011), 1218-1225
DOI: 10.1016/j.apradiso.2011.05.012
ISSN: 0969-8043
Long-Acting Lipidated Analogue of Human Pancreatic Polypeptide Is Slowly Released into Circulation
Bellmann-Sickert, K.; Elling, C. E.; Madsen, A. N.; Little, P. B.; Lundgren, K.; et al. (10 authors)
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Journal of Medicinal Chemistry 54(2011)8, 2658-2667
DOI: 10.1021/jm101357e
ISSN: 0022-2623
Synthesis, characterization and biological evaluation of [188Re(N)(cys∼)(PNP)]+/0 mixed-ligand complexes as prototypes for the development of 188Re(N)-based target-specific radiopharmaceuticals
Thieme, S.; Agostini, S.; Bergmann, R.; Pietzsch, J.; Pietzsch, H.-J.; et al. (9 authors)
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Nuclear Medicine and Biology 38(2011), 399-415
DOI: 10.1016/j.nucmedbio.2010.09.006
Synthesis and evaluation of 1,5-diaryl-substituted tetrazoles as novel selective cyclooxygenase-2 (COX-2) inhibitors
Al-Hourani, B. J.; Sharma, S. K.; Mane, J. Y.; Tuszynski, J.; Baracos, V.; et al. (9 authors)
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Bioorganic & Medicinal Chemistry Letters 21(2011), 1823-1826
DOI: 10.1016/j.bmcl.2011.01.057
ISSN: 0960-894X
Expression, purification and fluorine-18 radiolabeling of recombinant S100A4: a potential probe for molecular imaging of receptor for advanced glycation endproducts in vivo?
Wolf, S.; Haase-Kohn, C.; Lenk, J.; Hoppmann, S.; Bergmann, R.; et al. (7 authors)
- Amino Acids 41(2011), 809-820
A Novel Tetrabranched Neurotensin(8-13) Cyclam Derivative: Synthesis, 64Cu-Labeling and Biological Evaluation
Röhrich, A.; Bergmann, R.; Kretzschmann, A.; Noll, S.; Steinbach, J.; et al. (7 authors)
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Journal of Inorganic Biochemistry 105(2011), 821-832
DOI: 10.1016/j.jinorgbio.2011.02.011
Synthesis and biological evaluation of new [Tc(N)(PS)]-based mixed-ligand compounds useful in design of target-specific radiopharmaceuticas: the 2-methoxyphenylpiperazine dithiocarbamate derivatives as example
Bolzati, C.; Salvarese, N.; Carta, D.; Refosco, F.; Dolmella, A.; et al. (8 authors)
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Journal of Biological Inorganic Chemistry 16(2011), 137-155
DOI: 10.1007/s00775-010-0712-4
Automated radiosynthesis of the thiol-reactive labeling agent N-[6-(4-[18F]fluorobenzylidene)aminooxyhexyl]maleimide ([18F]FBAM)
Knieß, T.; Kuchar, M.; Pietzsch, J.
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Applied Radiation and Isotopes 69(2011), 1226-1230
DOI: 10.1016/j.apradiso.2011.03.043
2010
Modulation of Adrenal Aldosterone Release by Oxidative Modification of Low-Density Lipoprotein
Ansurudeen, I.; Pietzsch, J.; Graessler, J.; Ehrhart-Bornstein, M.; Saha, S.; et al. (7 authors)
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American Journal of Hypertension 23(2010)10, 1061-1068
DOI: 10.1038/ajh.2010.118
ISSN: 0895-7061
Identification of transport processes in bioirrigated muddy sediments by [18F]fluoride PET (Positron Emission Tomography)
Roskosch, A.; Lewandowski, J.; Bergmann, R.; Wilke, F.; Brenner, W.; et al. (6 authors)
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Applied Radiation and Isotopes 68(2010)6, 1094-1097
DOI: 10.1016/j.apradiso.2010.02.004
Comparison of the stability of Y-90-, Lu-177- and Ga-68- labeled human serum albumin microspheres (DOTA-HSAM)
Wunderlich, G.; Schiller, E.; Bergmann, R.; Pietzsch, H.-J.
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Nuclear Medicine and Biology 37(2010), 861-867
DOI: 10.1016/j.nucmedbio.2010.05.004
Preparation, 99mTc-labeling and biodistribution studies of a PNA oligomer containing a new ligand derivative of 2,2′-dipicolylamine
Gasser, G.; Jäger, K.; Zenker, M.; Bergmann, R.; Steinbach, J.; et al. (7 authors)
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Journal of Inorganic Biochemistry 104(2010), 1133-1140
DOI: 10.1016/j.jinorgbio.2010.06.011
Novel 99mTc '4 + 1' peptide conjugates: Tuning the biodistribution by variation of coligands
Künstler, J.-U.; Seidel, G.; Bergmann, R.; Gniazdowska, E.; Walther, M.; et al. (11 authors)
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European Journal of Medicinal Chemistry 45(2010), 3645-3655
DOI: 10.1016/j.ejmech.2010.05.010
Eph Receptors and Ephrin Ligands: Important Players in Angiogenesis and Tumor Angiogenesis
Mosch, B.; Reissenweber, B.; Neuber, C.; Pietzsch, J.
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Journal of Oncology 2010(2010), 135285
DOI: 10.1155/2010/135285
Cyclin-Dependent Kinase 4/6 (Cdk4/6) Inhibitors: Perspectives in Cancer Therapy and Imaging
Graf, F.; Mosch, B.; Koehler, L.; Bergmann, R.; Wuest, F.; et al. (6 authors)
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Mini-Reviews in Medicinal Chemistry 10(2010), 527-539
ISSN: 1389-5575
Synthesis of neurotensin(8-13)-phosphopeptide heterodimers via click chemistry
Richter, S.; Ramenda, T.; Bergmann, R.; Knieß, T.; Steinbach, J.; et al. (7 authors)
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Bioorganic & Medicinal Chemistry Letters 20(2010), 3306-3309
DOI: 10.1016/j.bmcl.2010.04.038
ISSN: 0960-894X
Radiosynthesis and radiopharmacological evaluation of cyclin-dependent kinase 4 (Cdk4) inhibitors
Koehler, L.; Graf, F.; Bergmann, R.; Steinbach, J.; Pietzsch, J.; et al. (6 authors)
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European Journal of Medicinal Chemistry 45(2010), 727-737
DOI: 10.1016/j.ejmech.2009.11.020
Scavenger receptors are associated with cellular interactions of S100A12 in vitro and in vivo
Hoppmann, S.; Steinbach, J.; Pietzsch, J.
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International Journal of Biochemistry & Cell Biology 42(2010), 651-661
DOI: 10.1016/j.biocel.2009.12.010
Effects of posture on regional pulmonary blood flow in rats as measured by PET
Richter, T.; Bergmann, R.; Pietzsch, J.; Közle, I.; Hofheinz, F.; et al. (8 authors)
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Journal of Applied Physiology 108(2010), 422-429
DOI: 10.1152/japplphysiol.91257.2008
Improved Multimodality Imaging Using Alginate Molding in Xenograft Tumor Models
Strobel, K.; Bergmann, R.; Meister, S.; van den Hoff, J.; Pietzsch, J.
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Journal of Magnetic Resonance Imaging 31(2010), 747-752
DOI: 10.1002/jmri.22090
2009
Fluorine-18 labeling of phosphopeptides: a potential approach for the evaluation of phosphopeptide metabolism in vivo.
Richter, S.; Bergmann, R.; Pietzsch, J.; Ramenda, T.; Steinbach, J.; et al. (6 authors)
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Biopolymers 92(2009)6, 479-488
DOI: 10.1002/bip.21263
Analysis of non-protein amino acids as specific markers of protein oxidation: the use of N(O,S)-ethoxycarbonyl ethyl ester and N(O,S)-ethoxycarbonyl trifluoroethyl ester derivatives and GC-MS
Pietzsch, J.; Pietzsch, F.-J.; Kopprasch, S.
- Trends in Chromatography 5(2009), 15-20
Radiolabelling of proteins with fluorine-18 via click chemistry
Ramenda, T.; Knieß, T.; Bergmann, R.; Steinbach, J.; Wüst, F.
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Chemical Communications 48(2009), 7521-7523
DOI: 10.1039/b916075b
ISSN: 1359-7345
Influence of irradiation on metabolism and metastatic potential of B16-F10 melanoma cells
Mosch, B.; Müller, K.; Steinbach, J.; Pietzsch, J.
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International Journal of Radiation Biology 85(2009)11, 1002-1012
DOI: 10.3109/09553000903258871
ISSN: 0955-3002
PET-Tracer für die onkologische Diagnostik: Welche radiomarkierten Substanzen sind relevant?
Knieß, T.; Steinbach, J.
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Onkologische Pharmazie 11(2009)4, 4-5
ISSN: 1437-8825
Autoradiographic studies of rhenium-188-hydroxyethylidine diphosphonate in normal skeleton and osteoblastic bone metastases in a rat model of metastatic prostate cancer
Liepe, K.; Geidel, H. H.; Bergmann, R.; Haase, M.; Runge, R.; et al. (6 authors)
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Nuclear Medicine Communications 30(2009), 693-699
DOI: 10.1097/MNM.0b013e32832cc23c
ISSN: 0143-3636
Comparison of [18F]FDG uptake and distribution with hypoxia and proliferation in FaDu human squamous cell carcinoma (hSCC) xenografts after single dose irradiation
Bruechner, K.; Bergmann, R.; Santiago, A.; Mosch, B.; Yaromina, A.; et al. (10 authors)
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International Journal of Radiation Biology 85(2009), 772-780
DOI: 10.1080/09553000903043067
ISSN: 0955-3002
Reduction of Arteriosclerotic Nanoplaque Formation and Size by n-3 Fatty Acids in Patients after Valvular Defect Operation
Koppe, C.; Rodriguez, M.; Winkler, K.; Pietzsch, J.; Neumann, K.; et al. (9 authors)
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Forschende Komplementärmedizin / Research in Complementary Medicine 16(2009), 237-245
DOI: 10.1159/000229786
Direct labelling of peptides with 2-[F-18]fluoro-2-deoxy-D-glucose ([F-18]FDG)
Wuest, F.; Hultsch, C.; Berndt, M.; Bergmann, R.
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Bioorganic & Medicinal Chemistry Letters 19(2009), 5426-5428
DOI: 10.1016/j.bmcl.2009.07.108
ISSN: 0960-894X
Radiosynthesis of New [90Y]-DOTA-Based Maleimide Reagents Suitable for the Prelabeling of Thiol-Bearing L-Oligonucleotides and Peptides
Schlesinger, J.; Fischer, C.; Közle, I.; Vonhoff, S.; Klussmann, S.; et al. (8 authors)
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Bioconjugate Chemistry 20(2009), 1340-1348
DOI: 10.1021/bc900095k
Fluorine-18 radiolabeling of native and oxidized proteins: An important tool in the pathophysiologists toolbox
Pietzsch, J.; Wuest, F.
- Chimica Oggi - Chemistry Today 27(2009), 12-14
Synthesis and radiopharmacological investigation of 3-[4-[18F]fluorobenzylidenyl]-indolin-2-one as possible tyrosine kinase inhibitor
Knieß, T.; Bergmann, R.; Kuchar, M.; Steinbach, J.; Wüst, F.
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Bioorganic & Medicinal Chemistry 17(2009), 7732-7742
DOI: 10.1016/j.bmc.2009.09.038
Fluorine-18-radiolabeled S100A12: a potential probe for functional characterization of inflammatory processes in vivo
Hoppmann, S.; Richter, S.; Steinbach, J.; Pietzsch, J.
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Inflammation Research 58(2009)Suppl. 2, S145-S146
ISSN: 1023-3830
Hexadentate Bispidine Derivatives as Versatile Bifunctional Chelate Agents for Copper(II) Radioisotopes
Juran, S.; Walther, M.; Stephan, H.; Bergmann, R.; Steinbach, J.; et al. (8 authors)
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Bioconjugate Chemistry 20(2009), 347-359
DOI: 10.1021/bc800461e
Synthesis and cyclooxygenase inhibition of various (aryl-1,2,3-triazole-1-yl)-methanesulfonylphenyl derivatives
Wuest, F.; Tang, X.; Knieß, T.; Pietzsch, J.; Suresh, M.
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Bioorganic & Medicinal Chemistry 17(2009), 1146-1151
DOI: 10.1016/j.bmc.2008.12.032
Radiosynthesis and radiopharmacological evaluation of [N-methyl-11C]Org 34850 as a glucocorticoid receptor (GR)-binding radiotracer
Wüst, F.; Knieß, T.; Henry, B.; Peeters, B. W. M. M.; Wiegerinck, P. H. G.; et al. (7 authors)
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Applied Radiation and Isotopes 67(2009), 308-312
DOI: 10.1016/j.apradiso.2008.10.014
Prediabetic and diabetic in vivo modification of circulating low density lipoprotein attenuates its stimulatory effect on adrenal mineralocorticoid secretion
Kopprasch, S.; Pietzsch, J.; Ansurudeen, I.; Graessler, J.; Krug, A. W.; et al. (7 authors)
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Journal of Endocrinology 200(2009), 45-52
DOI: 10.1677/JOE-08-0293
Validation of 99mTc-labeled "4+1" fatty acids for myocardial metabolism and flow imaging Part 2: Subcellular distribution
Mirtschink, P.; Stehr, S. N.; Walther, M.; Pietzsch, J.; Bergmann, R.; et al. (13 authors)
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Nuclear Medicine and Biology 36(2009), 845-852
DOI: 10.1016/j.nucmedbio.2009.06.003
Validation of 99mTc-labeled "4+1" fatty acids for myocardial metabolism and flow imaging Part 1: Myocardial extraction and biodistribution
Mirtschink, P.; Stehr, S. N.; Walther, M.; Pietzsch, J.; Bergmann, R.; et al. (13 authors)
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Nuclear Medicine and Biology 36(2009), 833-843
DOI: 10.1016/j.nucmedbio.2009.06.009
Cell cycle regulating kinase Cdk4 as a potential target for tumor cell treatment and tumor imaging
Graf, F.; Köhler, L.; Knieß, T.; Wüst, F.; Mosch, B.; et al. (6 authors)
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Journal of Oncology 2009(2009), 106378
DOI: 10.1155/2009/106378
Human S100A12: a novel key player in inflammation?
Pietzsch, J.; Hoppmann, S.
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Amino Acids 36(2009), 381-389
DOI: 10.1007/s00726-008-0097-7
ISSN: 0939-4451 (Print) 14
Systematic comparison of two novel thiol-reactive prosthetic groups for 18F labeling of peptides and proteins with the acylation agent succinimidyl-4-[18F]fluorobenzoate [18F]SFB
Wüst, F.; Köhler, L.; Berndt, M.; Pietzsch, J.
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Amino Acids 36(2009), 283-295
ISSN: 0939-4451
2008
Detailed Analysis Concerning the Biodistribution and Metabolism of Human Calcitonin-Derived Cell-Penetrating Peptides
Neundorf, I.; Rennert, R.; Franke, J.; Közle, I.; Bergmann, R.
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Bioconjugate Chemistry 19(2008)8, 1596-1603
DOI: 10.1021/bc800149f
Effects of pioglitazone and/or simvastatin on low density lipoprotein subfractions in non-diabetic patients with high cardiovascular risk: A sub-analysis from the PIOSTAT study
Leonhardt, W.; Pfützner, A.; Müller, J.; Pietzsch, J.; Forst, T.; et al. (8 authors)
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Atherosclerosis 201(2008), 155-162
DOI: 10.1016/j.atherosclerosis.2008.01.007
Synthesis and evaluation in vitro and in vivo of a 11C-labeled cyclooxygenase-2 (COX-2) inhibitor
Wüst, F.; Knieß, T.; Bergmann, R.; Pietzsch, J.
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Bioorganic & Medicinal Chemistry 16(2008), 7662-7670
DOI: 10.1016/j.bmc.2008.07.016
Yttrium-86-labelled human serum albumin microspheres: relation of surface structure with in vivo stability
Schiller, E.; Bergmann, R.; Pietzsch, J.; Noll, B.; Sterger, A.; et al. (8 authors)
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Nuclear Medicine and Biology 35(2008), 227-232
DOI: 10.1016/j.nucmedbio.2007.10.008
Synthesis and Application of [18F]FDG-maleimidehexyloxime ([18F]FDG-MHO): A [18F]FDG-based Prosthetic Group for the Chemoselective 18F-Labeling of Peptides and Proteins
Wüst, F.; Berndt, M.; Bergmann, R.; van den Hoff, J.; Pietzsch, J.
- Bioconjugate Chemistry 19(2008)6, 1202-1210
An 86Y-Labeled Mirror-Image Oligonucleotide: Influence of Y-DOTA Isomers on the Biodistribution in Rats
Schlesinger, J.; Közle, I.; Bergmann, R.; Tamburini, S.; Bolzati, C.; et al. (12 authors)
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Bioconjugate Chemistry 19(2008), 928-939
DOI: 10.1021/bc700453h
Facile synthesis of various nitro-substituted derivatives of semaxinib (SU 5416)
Knieß, T.; Kuchar, M.; Wüst, F.
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Synthetic Communications 38(2008), 3017-3022
DOI: 10.1080/00397910802044256
ISSN: 0039-7911 print/1532
Radiolabeled glucocorticoids as molecular probes for imaging brain glucocorticoid receptors by means of positron-emission-tomography (PET)
Steiniger, B.; Knieß, T.; Bergmann, R.; Pietzsch, J.; Wüst, F.
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Mini-Reviews in Medicinal Chemistry 8(2008)7, 728-739
ISSN: 1389-5575